CCL: How to select protein for docking



Hi Peter,

I understood that you want to ckeck with docking how your ligands work in some proteins (inhibitor, substrate, inert). (It's not enogh. You have to read about every protein to know them deeply). You should check the Protein Data Bank (PDB) http://www.rcsb.org/pdb/home/home.do">http://www.rcsb.org/pdb/home/home.do to download X-ray structures of different proteins and you can select a protein for docking taking into acount the active part of the protein (reading publications about that protein). But here I want to mention that in some cases the structure are not complete for docking. For example the ammonia-lyase structures have tetramer form, but in the PDB you can find them as dimer or two different dimer form. From here, after you know the real form of your protein and if this doesn't have the real form in the PDB you may build the real form in SwissPDBViewer program http://spdbv.vital-it.ch/">http://spdbv.vital-it.ch/.    It depends on your ligands too how they will fit  in the protein structure. You should check the electrophilic or nucleophilic properties at the ligands and in the active part (catalitic site) of the protein.
For docking you can use AutoDock http://autodock.scripps.edu/, FlexX http://www.biosolveit.de/flexx/ or other programs.
Hope this helps,
Good work,
Amalia
 
Amalia-Laura Seff
------------------------------------------------
PhD student
Babes-Bolyai University
Faculty of Chemistry and Chemical Engineering
Inorganic Chemistry Department
Molecular Modeling Laboratory 101
 
Adress: Arany János Str. no. 11
            Ro - 400028, Cluj-Napoca
tel: 40-264-593833/5772
      40-724752988
      36-702260428
fax: 40-264-590818
 



From: james peter jp07:+:sify.com <owner-chemistry[-]ccl.net>
To: "Seff, Amalia Laura -id#3td-" <slaurami[-]yahoo.com>
Sent: Sunday, June 14, 2009 3:14:11 PM
Subject: CCL: How to select protien for docking


Sent to CCL by: "james  peter" [jp07,sify.com]
Hi,
My work is on synthetic chemistry. I have synthesized a series of biologically activ compounds. just I want to perform protien ligand docking taking my molecules as ligand. My problem is how can I select a protien and from where I can download a protien.
I have read many tutorials describing method of docking taking an example protien and ligand. but my problem is how to select a protien from a wide list of protien structures and how to fit ligand structure into protine for docking. Please help me so that I can perform docking.
Thanking in advance
J.Peter



-= This is automatically added to each message by the mailing script =-
To recover the email address of the author of the message, please change
the strange characters on the top line to the [-] sign. You can also
look up the X-Original-From: line in the mail header.

E-mail to subscribers: CHEMISTRY[-]ccl.net or use:
      http://www.ccl.net/cgi-bin/ccl/send_ccl_message

E-mail to administrators: CHEMISTRY-REQUEST[-]ccl.net or use
      http://www.ccl.net/cgi-bin/ccl/send_ccl_message
      http://www.ccl.net/chemistry/sub_unsub.shtml

Before posting, check wait time at: http://www.ccl.net

Job: http://www.ccl.net/jobs
Conferences: http://server.ccl.net/chemistry/announcements/conferences/

Search Messages: http://www.ccl.net/chemistry/searchccl/index.shtml

If your mail bounces from CCL with 5.7.1 error, check:
      http://www.ccl.net/spammers.txt

RTFI: http://www.ccl.net/chemistry/aboutccl/instructions/