From owner-chemistry@ccl.net Sun Jan 9 19:07:00 2011 From: "Nancy nancy5villa]^[gmail.com" To: CCL Subject: CCL: Pioglitazone Tautomers Message-Id: <-43581-110109180916-14590-7E3+MJ2ZVD0/4BnZXj3h4Q#,#server.ccl.net> X-Original-From: Nancy Content-Type: multipart/mixed; boundary=20cf30433e32fd0028049971ef97 Date: Sun, 9 Jan 2011 18:09:03 -0500 MIME-Version: 1.0 Sent to CCL by: Nancy [nancy5villa.^^.gmail.com] --20cf30433e32fd0028049971ef97 Content-Type: multipart/alternative; boundary=20cf30433e32fd0021049971ef95 --20cf30433e32fd0021049971ef95 Content-Type: text/plain; charset=ISO-8859-1 Hi All, I am performing molecular docking and molecular dynamics simulations of the thiazolidinedione pioglitazone binding to the PPAR-gamma receptor protein (PDB ID: 1ZGY). The thiazolidinedione ring can exist in numerous different tautomeric states; I have attached a figure depicting several of them. Which tautomer would be dominant at the physiological pH of ~7.0? Also, are there any software programs that can predict which tautomer would be correct? Thanks in advance, Nancy --20cf30433e32fd0021049971ef95 Content-Type: text/html; charset=ISO-8859-1 Content-Transfer-Encoding: quoted-printable Hi All,

I am performing molecular docking and molecular dynamics sim= ulations of the thiazolidinedione pioglitazone binding to the PPAR-gamma re= ceptor protein (PDB ID: 1ZGY).=A0 The thiazolidinedione ring can exist in n= umerous different tautomeric states; I have attached a figure depicting sev= eral of them.=A0 Which tautomer would be dominant at the physiological pH o= f ~7.0?

Also, are there any software programs that can predict which tautomer w= ould be correct?

Thanks in advance,
Nancy


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